SCHEMBL8083650

SCHEMBL8083650

CCSC[C@@H](NC(c1ccccc1)c1ccccc1)C(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.45
PPARA Q07869 5/20 0.45
PPARD Q03181 2/20 0.43
CTSK P43235 4/20 0.42
CTSS P25774 3/20 0.42
MAPT P10636 4/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306604 0.82 MAPT (0.46) CTSKCTSSMAPTALDH1A1CTSL
SCHEMBL7317017 0.81 CTSK (0.47) CTSKCTSSMAPTALDH1A1KDM4E
SCHEMBL8083658 0.77 CTSK (0.46) CTSKCTSSMAPTALDH1A1GAA
SCHEMBL7316620 0.76 CTSK (0.57) CTSKCTSSALDH1A1PKMCYP2C19
SCHEMBL8075350 0.76 KMT2A (0.52) CTSKCTSSALDH1A1KDM4EHPGD
SCHEMBL8086793 0.76 KMT2A (0.52) CTSKCTSSALDH1A1KDM4EHPGD
SCHEMBL7307221 0.76 LMNA (0.41) MAPTALDH1A1GAAPKMHPGD
SCHEMBL7307182 0.75 CTSK (0.44) CTSKCTSSMAPTALDH1A1
SCHEMBL7304711 0.75 CTSK (0.44) CTSKCTSSMAPTALDH1A1
SCHEMBL6862901 0.72 ALDH1A1 (0.51) CTSKCTSSALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed