SCHEMBL7306975

SCHEMBL7306975

COc1ccc(C[C@H](N)CO)cc1OC(C)C

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.48
ALOX12 P18054 3/20 0.48
LDHA P00338 1/20 0.48
MMP1 P03956 1/20 0.47
CYP3A4 P08684 1/20 0.47
SIGMAR1 Q99720 7/20 0.46
FOS P01100 1/20 0.45
TTR P02766 1/20 0.45
JUN P05412 1/20 0.45
NR3C1 P04150 1/20 0.45
HSD17B1 P14061 1/20 0.45
HSD17B2 P37059 1/20 0.45
CA2 P00918 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ATM Q13315 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10776070 0.89 LDHA (0.58) ALOX15ALOX12LDHAMMP1CYP3A4
SCHEMBL7290411 0.89 LDHA (0.58) ALOX15ALOX12LDHAMMP1CYP3A4
SCHEMBL7298435 0.89 LDHA (0.58) ALOX15ALOX12LDHAMMP1CYP3A4
SCHEMBL13802900 0.81 CA2 (0.50) ALOX15ALOX12LDHACYP3A4FOS
SCHEMBL11695436 0.80 ALOX15 (0.66) ALOX15ALOX12MMP1CYP3A4FOS
SCHEMBL6344277 0.80 CYP3A4 (0.71) ALOX15ALOX12MMP1CYP3A4FOS
SCHEMBL4432280 0.79 MMP1 (0.53) LDHAMMP1CYP3A4FOSTTR
Hydrochloric Acid SCHEMBL11696571 0.79 ALOX15 (0.64) ALOX15ALOX12MMP1CYP3A4FOS
SCHEMBL24497200 0.78 LDHA (0.53) ALOX15ALOX12LDHACYP3A4FOS
SCHEMBL4748125 0.78 STAT3 (0.51) ALOX15ALOX12LDHACYP3A4CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490823-B1 Dihydro-isoquinoline derivates SANDOZ LTD (CH) 1996-11-13 EP disclosed
US-5177085-A DIHYDRO-ISOQUINOLINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE IN TREATING ASTHMA SANDOZ LTD. (CH) 1993-01-05 US disclosed
EP-0490823-A1 Dihydro-isoquinoline derivates SANDOZ LTD. (CH) 1992-06-17 EP disclosed