SCHEMBL7310236

SCHEMBL7310236

COc1ccc(SC2(CC(=O)O)CCCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.44
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
MMP12 P39900 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
EP300 Q09472 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NPC1 O15118 2/20 0.38
TP53 P04637 1/20 0.38
PDE4B Q07343 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305235 0.85 MMP1 (0.47) MMP2MMP9MMP12NPC1TP53
SCHEMBL7303726 0.84 ALDH1A1 (0.44) ALDH1A1MAPTMEN1KMT2A
SCHEMBL7307399 0.83 ALDH1A1 (0.43) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL6658727 0.79 ADAM17 (0.47) ALDH1A1MMP2MMP9KMT2A
SCHEMBL618046 0.78 FFAR1 (0.41) HSD11B1ALDH1A1HPGDTSHRCYP2C19
SCHEMBL7303615 0.77 SCN5A (0.49) TSHRMMP2MMP9CYP2C19NPC1
SCHEMBL364190 0.73 HSD11B1 (0.65) HSD11B1ALDH1A1HPGDTSHRCYP3A4
SCHEMBL9637668 0.71 ALDH1A1 (0.40) ALDH1A1HPGDTSHR
SCHEMBL7306362 0.71 MMP1 (0.49) ALDH1A1MMP2MMP9MMP12MAPT
SCHEMBL11619962 0.71 SLC6A4 (0.45) ALDH1A1HPGDCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed