SCHEMBL7227670

SCHEMBL7227670

CC(C)(C)OC(=O)N1CCN(CCCN2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.41
CHRM1 P11229 2/20 0.41
STAT3 P40763 1/20 0.38
GPR119 Q8TDV5 6/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TLR8 Q9NR97 1/20 0.35
EPHX2 P34913 4/20 0.35
ACKR3 P25106 3/20 0.35
CHRM4 P08173 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7228352 0.98 CHRM2 (0.41) CHRM2CHRM1STAT3GPR119MAPK1
SCHEMBL7236582 0.94 CHRM2 (0.38) CHRM2CHRM1STAT3GPR119ACKR3
SCHEMBL7310460 0.86 SIGMAR1 (0.34) CHRM2CHRM1STAT3MAPK1L3MBTL1
SCHEMBL7313917 0.85 SIGMAR1 (0.34) CHRM2CHRM1STAT3MAPK1L3MBTL1
SCHEMBL7316915 0.82 MAPK1 (0.45) MAPK1L3MBTL1
SCHEMBL7313718 0.81 SIGMAR1 (0.31) MAPK1L3MBTL1
SCHEMBL7306386 0.80 MAPK1 (0.47) MAPK1L3MBTL1
SCHEMBL7310863 0.79 MAPK1 (0.40) MAPK1L3MBTL1
SCHEMBL7306591 0.78 TP53 (0.42) GPR119EPHX2
SCHEMBL7313885 0.77 GPR119 (0.38) GPR119MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed