SCHEMBL7312649

SCHEMBL7312649

Nc1cc(-c2cccc(-c3ccccc3)c2)n[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.51
AURKA O14965 1/20 0.51
THRB P10828 1/20 0.51
CASP1 P29466 1/20 0.51
TTK P33981 1/20 0.51
AURKB Q96GD4 1/20 0.51
INCENP Q9NQS7 1/20 0.51
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
PDE2A O00408 1/20 0.47
ADORA3 P0DMS8 1/20 0.46
PRMT5 O14744 1/20 0.44
POLB P06746 2/20 0.43
RAB9A P51151 1/20 0.43
TP53 P04637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 1/20 0.42
DAO P14920 1/20 0.42
JAK2 O60674 2/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1392639 0.90 ADORA3 (0.56) MAPTAURKATHRBCASP1TTK
SCHEMBL28025294 0.83 POLB (0.48) MAPTAURKATHRBCASP1TTK
SCHEMBL2823296 0.83 IDO1 (0.47) MAPTAURKATHRBCASP1TTK
SCHEMBL11245286 0.77 CYP1A2 (0.63) AURKATTKAURKBINCENPPDE3B
SCHEMBL11242864 0.75 PDE3B (0.61) MAPTAURKATHRBCASP1TTK
SCHEMBL17775678 0.74 RAB9A (0.78) MAPTADORA3POLBRAB9ATP53
SCHEMBL17279909 0.74 POLB (0.71) MAPTADORA3POLBRAB9ATP53
SCHEMBL11293296 0.72 PIN1 (0.54) MAPTPDE3BPDE3APDE2APRMT5
Hydrochloric Acid SCHEMBL11246455 0.72 PDE3B (0.58) MAPTAURKATHRBCASP1TTK
SCHEMBL1754735 0.72 POLB (0.57) MAPTAURKBADORA3POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394998-A1 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3-yl)-biphenyl derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-12-14 EP disclosed