SCHEMBL7320271

SCHEMBL7320271

Cc1ccc(S(=O)(=O)N(C(=O)[C@H]2NCCS2)[C@@H](Cc2ccc(OCCCN(C)C)cc2)C(=O)O)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.37
ITGA2B P08514 4/20 0.37
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CACNA1B Q00975 2/20 0.34
POLB P06746 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA5 P08648 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
ADAM17 P78536 1/20 0.34
PKM P14618 1/20 0.34
LMNA P02545 1/20 0.34
PPARG P37231 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314611 0.86 ITGB3 (0.35) ITGB3ITGA2BKMT2AMEN1ALDH1A1
SCHEMBL7069676 0.84 ADAMTS5 (0.43) KMT2AALDH1A1POLBMMP9CNR2
SCHEMBL7326742 0.83 ITGB3 (0.37) ITGB3ITGA2BKMT2AMEN1ALDH1A1
SCHEMBL7319946 0.82 KMT2A (0.35) ITGB3ITGA2BKMT2AMEN1ALDH1A1
SCHEMBL3856501 0.79 TAS2R14 (0.35) ITGB3ITGA2BALDH1A1ITGB1ITGAV
SCHEMBL7318412 0.78 ALDH1A1 (0.37) KMT2AMEN1ALDH1A1POLBLTB4R
SCHEMBL7069725 0.77 LMNA (0.40) ALDH1A1POLBLMNA
SCHEMBL7316484 0.76 F2 (0.33) ITGB3ITGA2BKMT2AMEN1ALDH1A1
SCHEMBL3850724 0.76 P2RX7 (0.33) ALDH1A1MMP13LMNA
SCHEMBL7385520 0.76 TAS2R14 (0.41) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492421-B1 BINDING VERY LATE ANTIGEN-4; INFLAMMATORY DISEASES SUCH AS ASTHMA, ALZHEIMER'S DISEASE, ATHEROSCLEROSIS, AIDS, DEMENTIA, DIABETES, INFLAMMATORY BOWEL DISEASE, RHEUMATOID ARTHRITIS, TISSUE TRANSPLANTATION, TUMOR METASTASIS, MYOCARDIAL ISCHEMIA ATHENA NEUROSCIENCES, INC. 2002-12-10 US claimed
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-6492421-B1 BINDING VERY LATE ANTIGEN-4; INFLAMMATORY DISEASES SUCH AS ASTHMA, ALZHEIMER'S DISEASE, ATHEROSCLEROSIS, AIDS, DEMENTIA, DIABETES, INFLAMMATORY BOWEL DISEASE, RHEUMATOID ARTHRITIS, TISSUE TRANSPLANTATION, TUMOR METASTASIS, MYOCARDIAL ISCHEMIA ATHENA NEUROSCIENCES, INC. 2002-12-10 US disclosed