SCHEMBL7323478

SCHEMBL7323478

C=CCN(CC=C)C1CCC(O)CC1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2363531 0.88 SIGMAR1 (0.35) LSSSIGMAR1OPRM1OPRD1OPRK1
SCHEMBL12473169 0.88 SHBG (0.32) OPRM1OPRD1OPRK1
SCHEMBL14984946 0.78 OPRM1 (0.34) SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL2163192 0.78 ALDH1A1 (0.38) SIGMAR1
SCHEMBL30750 0.76 ALDH1A1 (0.41) SIGMAR1
Fluoride SCHEMBL9620616 0.74 ALDH1A1 (0.40) SIGMAR1
Hydrochloric Acid SCHEMBL2957420 0.74 ALDH1A1 (0.40) SIGMAR1
Ammonia Solution, Strong SCHEMBL17439397 0.74 ALDH1A1 (0.40) SIGMAR1
SCHEMBL12403631 0.74
SCHEMBL7269723 0.73 SIGMAR1 (0.31) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4886812-A REGULATING DOPAMINE CONCENTRATION; PARKINSON DISEASE, HYPOTENSIVE AGENT, SCHIZOPHRENIA DR. KARL THOMAE GMBH (DE) 1989-12-12 US disclosed
US-4843086-A HYPOTENSIVE AGENTS, SCHIZOPHRENIA, PARKINSON'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1989-06-27 US disclosed
US-4731374-A PARKINSON*S DISEASE DR. KARL THOMAE GMBH (DE) 1988-03-15 US disclosed
EP-0186087-A1 Tetrahydro-benzothiazoles, their production and their use as intermediates or drugs Dr. Karl Thomae GmbH (DE) 1986-07-02 EP disclosed