SCHEMBL7326237

SCHEMBL7326237

Cc1c(CNC(=O)c2cn3c4c(cccc24)CCC3C)ncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 2/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CNR1 P21554 2/20 0.33
ELANE P08246 6/20 0.32
CCR1 P32246 3/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334672 0.85 MTNR1A (0.41) HPGDSMN1; SMN2
SCHEMBL7326609 0.79 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DKDM4E
Hydrochloric Acid SCHEMBL9730335 0.78 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL7329638 0.70 KDM4E (0.57) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6334232 0.66 KDM4E (0.44) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL3965154 0.66 KDM4E (0.67) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL3966675 0.66 KDM4E (0.67) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL7318822 0.65 KDM4E (0.44) KDM4EHPGDSMN1; SMN2
SCHEMBL7274096 0.65 MEN1 (0.37) KDM4E
SCHEMBL9789206 0.64 MCL1 (0.35) KDM4EHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5102901-A 5-hydroxytrypamine receptor antaonists DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1992-04-07 US disclosed
EP-0393766-A2 New 3-N substituted carbamoyl-indole derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-10-24 EP disclosed