SCHEMBL7327775

SCHEMBL7327775

Cc1cc(C2(C(=O)OC(C)(C)C)CCNCC2)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.43
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
POLB P06746 1/20 0.36
CASP6 P55212 1/20 0.36
AKR1B10 O60218 1/20 0.35
AKR1C4 P17516 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326235 0.78 OPRM1 (0.56) OPRM1
SCHEMBL654834 0.72 DRD2 (0.54) OPRM1HDAC3HDAC1HDAC2HDAC6
SCHEMBL29510643 0.71 MIF (0.38) AKR1B10AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL31173465 0.70 ASIC3 (0.42)
SCHEMBL3174988 0.69 OPRM1 (0.34) OPRM1
SCHEMBL14258104 0.69 OPRM1 (0.49) OPRM1
SCHEMBL7613755 0.68 ALDH1A1 (0.48) OPRM1POLBAKR1C1
SCHEMBL7924071 0.68 OPRM1 (0.43) OPRM1
SCHEMBL14161293 0.67 HSD11B1 (0.50) OPRM1
SCHEMBL29510626 0.67 OPRM1 (0.47) OPRM1POLBAKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376506-B1 REACTING SULFAMOYL OXAZOLIDONE WITH (1,2,3,4)-TETRAHYDRO-BETA-CARBOLINE TO FORM INHIBITOR; USED TO TREAT ARTHRITIS, OSTEOPOROSIS, PERIODONTAL DISEASE, CARDIOVASCULAR DISEASES, MULTIPLE SCLEROSIS, AND TUMORS SYNTEX (U.S.A.) LLC 2002-04-23 US disclosed