SCHEMBL7328239

SCHEMBL7328239

c1ccc(COc2ccnc(-c3ccc4[nH]ccc4c3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.49
NPC1 O15118 1/20 0.48
CYP17A1 P05093 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
XDH P47989 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
ALKBH1 Q13686 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
BACE1 P56817 1/20 0.40
MAP3K11 Q16584 1/20 0.40
GLO1 Q04760 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
CTNNB1 P35222 2/20 0.38
WNT3A P56704 2/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA10 Q9GZZ6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868720 0.79 DYRK3 (0.51) NPC1CYP17A1CYP11B1CYP11B2S1PR1
SCHEMBL7464319 0.78 PDE5A (0.50) XDHALKBH1L3MBTL1
SCHEMBL3901006 0.77 NPC1 (0.64) ENPP2NPC1CYP17A1CYP11B1CYP11B2
SCHEMBL18828552 0.75 NPC1 (0.59) NPC1CYP17A1CYP11B1CYP11B2S1PR1
SCHEMBL5103334 0.73 GABRG2 (0.56) ENPP2NPC1LOXL2BACE1CYP19A1
SCHEMBL329575 0.73 ALOX5 (0.62) ENPP2NPC1NSD2ABL1PPARG
SCHEMBL6669227 0.72 ENPP2 (0.48) ENPP2NPC1CYP17A1CYP11B1CYP11B2
Pyridine SCHEMBL28518713 0.72 ALOX5 (0.53) ENPP2NPC1CYP17A1CYP11B1CYP11B2
SCHEMBL30488441 0.72 GRM5 (0.43) ENPP2LOXL2NSD2ABL1PPARG
SCHEMBL5364336 0.72 GRM5 (0.43) ENPP2LOXL2NSD2ABL1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed