SCHEMBL7328319

SCHEMBL7328319

C=C(c1ccccc1OCCCNC(C)(C)C)c1cccc2[nH]ccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 1/20 0.47
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
HTR1A P08908 7/20 0.44
SLC6A4 P31645 3/20 0.43
GAA P10253 1/20 0.40
MCL1 Q07820 1/20 0.39
DHPS P49366 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327839 0.87 HTR1B (0.47) HTR1BDRD2DRD4DRD3HTR1A
SCHEMBL9449999 0.83 HTR1B (0.48) HTR1BDRD2DRD4DRD3HTR1A
SCHEMBL9450175 0.83 DRD2 (0.43) HTR1BDRD2DRD4DRD3HTR1A
SCHEMBL7333081 0.82 ADRB2 (0.54) HTR1BDRD4DRD3HTR1A
SCHEMBL7325339 0.82 HDAC1 (0.41) HTR1BDRD2DRD4DRD3HTR1A
Benzoic Acid SCHEMBL9449941 0.82 DRD2 (0.43) HTR1BDRD2DRD4DRD3HTR1A
SCHEMBL9130336 0.81 DHPS (0.50) HTR1BDRD2DRD4DRD3GAA
Hydrochloric Acid SCHEMBL9130882 0.81 DHPS (0.48) HTR1BDRD2DRD4DRD3HTR1A
SCHEMBL10502612 0.80 HTR1A (0.46) HTR1BDRD2DRD4DRD3HTR1A
Hydrochloric Acid SCHEMBL10572848 0.79 HTR1A (0.46) HTR1BDRD2DRD4DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0395528-B1 4-Phenylmethyl-1H-indole derivatives, process and intermediates for their preparation, their use as medicines and compositions containing them ROUSSEL UCLAF (FR) 1995-07-05 EP claimed
US-5086070-A 4-BENZYL-1H-INDOLES AND ANTI-ARRTHYMIC USE THEREOF ROUSSEL UCLAF (FR) 1992-02-04 US claimed
US-5182282-A Antiarrhythmia agents ROUSSEL UCLAF (FR) 1993-01-26 US disclosed
US-5086070-A 4-BENZYL-1H-INDOLES AND ANTI-ARRTHYMIC USE THEREOF ROUSSEL UCLAF (FR) 1992-02-04 US disclosed