SCHEMBL7328372

SCHEMBL7328372

Cc1cccc(-c2c[n+]3ccn(C)c3c(=O)[nH]2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
TDP2 O95551 1/20 0.35
MEN1 O00255 1/20 0.34
CASP3 P42574 1/20 0.34
KMT2A Q03164 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
XDH P47989 1/20 0.34
ALDH1A1 P00352 2/20 0.34
PBRM1 Q86U86 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
NPY5R Q15761 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7330447 0.86 BRD4 (0.41) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL7327728 0.85 TNKS (0.37) ALDH1A1KDM4EMAPTADORA3
SCHEMBL7327598 0.84 TNKS (0.41) NPC1RAB9AMEN1KMT2AL3MBTL1
SCHEMBL7331031 0.82 MAPT (0.48) NPC1MEN1KMT2AALDH1A1MAPT
SCHEMBL7329537 0.77 ALDH1A1 (0.37) NPC1RAB9AMEN1KMT2AL3MBTL1
SCHEMBL7331334 0.76 BRD4 (0.36) NPC1RAB9ATDP2ALDH1A1KDM4E
SCHEMBL7337599 0.74 TNKS (0.39) TDP2ALDH1A1KDM4E
SCHEMBL7338197 0.73 CTSV (0.35) MEN1KMT2AL3MBTL1ALDH1A1KDM4E
SCHEMBL7328378 0.72 TNKS (0.38) NPC1RAB9ATDP2MEN1CASP3
SCHEMBL17016650 0.67 PARP1 (0.45) NPC1RAB9AL3MBTL1XDHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726900-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS Aventis Pharma S.A. (FR) 1996-08-21 EP disclosed
WO-1995012594-A1 7H-IMIDAZO(1,2-a)PYRAZINE-8-ONE NMDA RECEPTOR ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-05-11 WO disclosed