SCHEMBL7329563

SCHEMBL7329563

COP(=O)(OC)[C@@H](CCN1C(=O)c2cccc3c(Br)ccc(c23)C1=O)NC(CC(C)C)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 5/20 0.45
ALDH1A1 P00352 2/20 0.44
POLB P06746 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
PABPC1 P11940 1/20 0.44
KMT2A Q03164 1/20 0.44
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
TLR9 Q9NR96 1/20 0.43
MMP1 P03956 10/20 0.42
MMP9 P14780 10/20 0.42
MMP3 P08254 8/20 0.42
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9349379 0.88 CYP1B1 (0.46) CYP1B1MMP1MMP9MMP3
SCHEMBL7329953 0.88 MMP1 (0.50) POLBKDM4EMEN1KMT2AMMP1
SCHEMBL7323303 0.87 MMP9 (0.52) POLBMEN1KMT2AMMP1MMP9
SCHEMBL7323291 0.87 MMP9 (0.52) POLBMEN1KMT2AMMP1MMP9
SCHEMBL7323279 0.87 MMP9 (0.52) POLBMEN1KMT2AMMP1MMP9
SCHEMBL7329042 0.81 MMP1 (0.47) CYP1B1MMP1MMP9MMP3
SCHEMBL6417587 0.76 MMP1 (0.47) CYP1B1MMP1MMP9MMP3
SCHEMBL7356722 0.76 ECE1 (0.49)
SCHEMBL23752622 0.75 KEAP1 (0.71) CYP1B1ALDH1A1POLBKDM4EMEN1
SCHEMBL7322384 0.74 MMP1 (0.54) MMP1MMP9MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612324-A1 PHOSPHONOPEPTIDES WITH COLLAGENASE INHIBITING ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1994-08-31 EP disclosed
WO-1993009136-A1 PHOSPHONOPEPTIDES WITH COLLAGENASE INHIBITING ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1993-05-13 WO disclosed