SCHEMBL7329772

SCHEMBL7329772

CC(C)(C)OC(=O)N(N)Cc1cncs1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.40
PARP15 Q460N3 1/20 0.38
PARP10 Q53GL7 1/20 0.38
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
LMNA P02545 3/20 0.33
GPR119 Q8TDV5 1/20 0.33
ACACB O00763 1/20 0.32
USP30 Q70CQ3 1/20 0.32
HTT P42858 2/20 0.32
SLC6A3 Q01959 2/20 0.32
CTSK P43235 1/20 0.31
ACLY P53396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325509 0.74 GPR119 (0.34) GPR119ACACB
SCHEMBL19475116 0.74 RAB9A (0.40) TRPM8PARP15PARP10RAB9ANPC1
SCHEMBL9933949 0.72 NPC1 (0.44) RAB9ANPC1SMN1; SMN2TDP1LMNA
SCHEMBL8336083 0.72 CYP17A1 (0.44) RAB9ASMN1; SMN2LMNAGPR119HTT
SCHEMBL7328855 0.71 KDR (0.31)
SCHEMBL3064090 0.71 HRH4 (0.39) TRPM8RAB9ANPC1LMNAHTT
SCHEMBL7332333 0.70 RIPK1 (0.51) TRPM8RAB9ASMN1; SMN2LMNAHTT
SCHEMBL9933946 0.70 PAX8 (0.38) TRPM8GPR119USP30
SCHEMBL2061999 0.68 AKT1 (0.50) RAB9ANPC1HTT
SCHEMBL4832991 0.68 GSTO1 (0.34) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990135-A FOR TREATING A RETROVIRAL INFECTION SUCH AS HIV INFECTION; FOR EXAMPLE 5S-N-((2-PYRIDINYL)METHOXYCARBONYL)VALINYLAMINO-2-((N-3 -PYRIDINYL)METHOXYCARBONYL)AMINO-4S-HYDROXY-1,6-DIPHENYL-2-AZAHEXANE AND OTHER COMPOUNDS OF GIVEN FORMULA ABBOTT LABORATORIES (US) 1999-11-23 US disclosed
US-5631376-A PEPTIDE DERIVATIVES FOR TREATMENT OF AIDS ABBOTT LABORATORIES (US) 1997-05-20 US disclosed
US-5621109-A OXAZOLE/THIAZOLE DERIVATIVES OF HYDROXYMETHYL HYDRAZONES; SIDE EFFECT REDUCTION ABBOTT LABORATORIES (US) 1997-04-15 US disclosed
US-5461067-A For HIV infections ABBOTT LABORATORIES (US) 1995-10-24 US disclosed
WO-1994019332-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1994-09-01 WO disclosed