SCHEMBL7329778

SCHEMBL7329778

CN(CCc1ccc(O)cc1)C(=O)c1ccc(C#N)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 1/20 0.65
NSD2 O96028 2/20 0.58
MCHR1 Q99705 2/20 0.49
PDK1 Q15118 2/20 0.48
PDK2 Q15119 1/20 0.48
PDK3 Q15120 1/20 0.48
PDK4 Q16654 1/20 0.48
CYP19A1 P11511 2/20 0.48
MLYCD O95822 2/20 0.48
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
CA12 O43570 1/20 0.44
CA2 P00918 1/20 0.44
CA3 P07451 1/20 0.44
CA6 P23280 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796753 0.86 NSD2 (0.77) ESRRGNSD2PDK1PDK2PDK3
SCHEMBL5317404 0.79 NSD2 (0.58) NSD2PDK2MLYCDCA2MEN1
SCHEMBL6794239 0.75 CA2 (0.52) NSD2PDK1PDK2PDK3PDK4
SCHEMBL14357352 0.75 LTB4R (0.52) NSD2MLYCDTSHRRAB9ANPC1
SCHEMBL10355508 0.75 CA2 (0.73) CYP19A1ESR1ESR2CA12CA2
SCHEMBL5318145 0.74 NSD2 (0.60) NSD2PDK1PDK2PDK3PDK4
SCHEMBL23015300 0.73 NSD2 (1.00) NSD2MCHR1PDK1PDK2PDK3
SCHEMBL6799435 0.73 MEN1 (0.72) NSD2PDK1PDK2PDK3PDK4
SCHEMBL5414969 0.73 NSD2 (0.52) NSD2PDK2MLYCDCA2MEN1
SCHEMBL21996676 0.72 PPARA (0.43) ESRRGNSD2CYP19A1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP disclosed
EP-0381033-A1 Carboxylic-acid and sulphonic-acid amides F. HOFFMANN-LA ROCHE AG (CH) 1990-08-08 EP disclosed