SCHEMBL7340682

SCHEMBL7340682

CS(=O)(=O)c1cccc(CC(NC(=O)CNC(=O)c2cccc(NC=NN)c2)C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
HSD17B10 Q99714 1/20 0.47
ITGB2 P05107 2/20 0.41
ICAM1 P05362 2/20 0.41
ITGAL P20701 2/20 0.41
ITGB1 P05556 6/20 0.40
ITGA4 P13612 1/20 0.40
CTSB P07858 2/20 0.39
GPR132 Q9UNW8 1/20 0.39
ITGB3 P05106 4/20 0.39
ITGAV P06756 4/20 0.39
ITGA2B P08514 2/20 0.39
ITGB5 P18084 2/20 0.39
CTSV O60911 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
CA2 P00918 2/20 0.39
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6775970 0.89 GPR132 (0.49) ITGB1GPR132ITGB3ITGAVITGA2B
SCHEMBL6772224 0.87 CTSV (0.50) ITGB1CTSBGPR132ITGB3ITGAV
SCHEMBL7838300 0.87 ITGB3 (0.51) ITGB1CTSBGPR132ITGB3ITGAV
SCHEMBL6773776 0.86 CTSB (0.43) GAAITGB1CTSBGPR132ITGB3
SCHEMBL7345772 0.86 GPR132 (0.39) ALDH1A1ITGB1CTSBGPR132ITGB3
SCHEMBL6778268 0.85 GPR139 (0.44) ITGB1CTSBGPR132ITGB3ITGAV
SCHEMBL3051751 0.84 GPR139 (0.44) ITGB1CTSBGPR132ITGB3ITGAV
SCHEMBL7823171 0.84 ITGB3 (0.50) ITGB1GPR132ITGB3ITGAVITGA2B
SCHEMBL7339636 0.84 GPR132 (0.50) ALDH1A1GPR132SMN1; SMN2GPR139
SCHEMBL6778084 0.84 GPR139 (0.45) ITGB1ITGA4CTSBGPR132ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed