SCHEMBL7340893

SCHEMBL7340893

C[C@@H](C(=O)O)N1CCCC[C@H](N2C(=O)c3ccccc3C2=O)C1=O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HTT P42858 1/20 0.44
XIAP P98170 2/20 0.43
ACE P12821 1/20 0.43
POLB P06746 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CHRM2 P08172 1/20 0.38
OPRM1 P35372 1/20 0.38
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
IKZF3 Q9UKT9 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7342538 0.81 ALDH1A1 (0.52) ALDH1A1HTTPOLBLMNAKMT2A
SCHEMBL12589545 0.81 ALDH1A1 (0.52) ALDH1A1HTTPOLBLMNAKMT2A
SCHEMBL7501387 0.79 ALOX15 (0.43) ALDH1A1HTTXIAPLMNAKMT2A
SCHEMBL8212856 0.79 ALOX15 (0.43) ALDH1A1HTTXIAPLMNAKMT2A
SCHEMBL12589543 0.75 ACE (0.48) ALDH1A1ACEPOLBKMT2AL3MBTL1
SCHEMBL7063281 0.74 LMNA (0.38) ALDH1A1HTTLMNAKMT2AL3MBTL1
SCHEMBL8358951 0.72 ACE (0.49) XIAPACE
SCHEMBL10793023 0.71 ACE (0.51) XIAPACETSHRTDP1
SCHEMBL10793019 0.71 ACE (0.51) XIAPACETSHRTDP1
SCHEMBL7340816 0.71 ACE (0.51) XIAPACETSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0599444-B1 Dual action inhibitors SQUIBB & SONS INC (US) 1998-01-28 EP disclosed
US-5654294-A CARDIOVASCULAR DISORDERS BRISTOL-MYERS SQUIBB (US) 1997-08-05 US disclosed
EP-0783002-A2 Dual action inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-07-09 EP disclosed
US-5646276-A ANGIOTENSIN CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE INHIBITORS; CARDIOVASCULAR DISORDERS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-08 US disclosed
US-5552397-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-09-03 US disclosed
EP-0599444-A1 Dual action inhibitors E.R. SQUIBB & SONS, INC. (US) 1994-06-01 EP disclosed