SCHEMBL7344613

SCHEMBL7344613

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccsc1.c1ccc2c(c1)CNC2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.61
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 3/20 0.54
HSD17B10 Q99714 3/20 0.54
HPGD P15428 2/20 0.54
CACNA1B Q00975 1/20 0.54
ADORA2B P29275 3/20 0.53
POLB P06746 2/20 0.53
CASP1 P29466 1/20 0.51
PKM P14618 1/20 0.50
HIF1A Q16665 3/20 0.49
MEN1 O00255 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
KMT2A Q03164 2/20 0.49
MAPT P10636 2/20 0.49
TSHR P16473 2/20 0.49
LMNA P02545 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3002791 0.84 ADORA2B (0.67) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL10744169 0.82 ALDH1A1 (0.57) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL3033425 0.82 HSD17B10 (0.69) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7344610 0.81 HSD17B10 (0.52) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7341782 0.81 CACNA1D (0.67) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7347764 0.81 ADORA3 (0.64) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7345498 0.81 ADORA3 (0.64) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7343711 0.81 ADORA3 (0.64) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7349302 0.81 ADORA3 (0.64) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7344616 0.80 CACNA1B (0.49) ADORA3KDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed