SCHEMBL7353583

SCHEMBL7353583

CCCCS(=O)(=O)N(CC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C(CCC(C)C)NC(=O)NC(C)(C)C)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.37
CTSD P07339 8/20 0.37
REN P00797 2/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
PSMB5 P28074 2/20 0.33
BCHE P06276 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8899924 0.92 BACE1 (0.36) BACE1CTSDRENBCHE
SCHEMBL7360719 0.88 BACE1 (0.36) BACE1CTSDRENBACE2
SCHEMBL7353577 0.84 REN (0.34) BACE1CTSDRENOPRM1OPRD1
SCHEMBL8897548 0.83 BACE1 (0.33) BACE1CTSDREN
SCHEMBL7476233 0.82 SPPL2A (0.38) BACE1CTSD
SCHEMBL8840299 0.80 BACE1 (0.40) BACE1RENBCHE
SCHEMBL8606263 0.78 BACE1 (0.35) BACE1REN
SCHEMBL7360716 0.78 BACE1 (0.36) BACE1CTSDREN
SCHEMBL8897311 0.74 REN (0.38) RENBCHE
SCHEMBL8897322 0.74 REN (0.38) RENBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614522-A SULFONAMIDE AND UREA-CONTAINING HYDROXYETHYLAMINE COMPOUNDS G.D. SEARLE & CO. (US) 1997-03-25 US disclosed
EP-0558673-A1 RETROVIRAL PROTEASE INHIBITORS. MONSANTO CO (US) 1993-09-08 EP disclosed
WO-1992008699-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed