SCHEMBL7353587

SCHEMBL7353587

O=C(O)c1cccc(Cn2c(=O)c(=O)[nH]c3ccc([N+](=O)[O-])cc32)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.52
FEN1 P39748 1/20 0.49
TP53 P04637 1/20 0.46
NOX4 Q9NPH5 1/20 0.46
PKM P14618 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GRIK1 P39086 3/20 0.44
GRIK2 Q13002 3/20 0.44
GRIK3 Q13003 3/20 0.44
GRIK4 Q16099 3/20 0.44
GRIK5 Q16478 3/20 0.44
CCR2 P41597 1/20 0.44
GRIA1 P42261 2/20 0.43
GRIA2 P42262 2/20 0.43
GRIA3 P42263 2/20 0.43
GRIA4 P48058 2/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358171 0.92 FEN1 (0.49) PGRFEN1TP53NOX4PKM
SCHEMBL7352784 0.88 PGR (0.49) PGRFEN1NOX4GRIK1GRIK2
SCHEMBL7353213 0.88 PGR (0.46) PGRFEN1NOX4ALDH1A1KMT2A
SCHEMBL7356210 0.85 TP53 (0.52) FEN1TP53NOX4PKMMAPK1
SCHEMBL7359747 0.82 PGR (0.45) PGRNOX4GRIK1GRIK2GRIK3
SCHEMBL7349906 0.80 NOX4 (0.45) FEN1NOX4CCR2ALDH1A1KMT2A
SCHEMBL12822268 0.80 PKM (0.48) PGRFEN1TP53NOX4PKM
SCHEMBL7352345 0.80 CCR2 (0.46) FEN1NOX4GRIK1GRIK2GRIK3
SCHEMBL9556876 0.79 PGR (0.50) PGRNOX4GRIK1GRIK2GRIK3
SCHEMBL9093246 0.79 GRIA1 (0.58) GRIK1GRIK2GRIK3GRIK4GRIK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed