SCHEMBL7354891

SCHEMBL7354891

N#Cc1ccc(NC(=O)Cn2ccc3cc(N)ccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 1/20 0.52
RORC P51449 9/20 0.48
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 5/20 0.47
TSHR P16473 3/20 0.47
HSD17B10 Q99714 3/20 0.47
HPGD P15428 2/20 0.47
GLA P06280 1/20 0.47
HTT P42858 1/20 0.47
USP2 O75604 1/20 0.46
POLB P06746 1/20 0.46
NPY5R Q15761 1/20 0.43
KCNA5 P22460 1/20 0.42
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357276 0.82 KRAS (0.52) RORCKDM4EALDH1A1TSHRHSD17B10
SCHEMBL20941549 0.74 SAE1 (0.54) KDM4EALDH1A1TSHRHTTPOLB
SCHEMBL8248060 0.73 NTSR1 (0.55) NTSR1
SCHEMBL3465527 0.72 KMT2A (0.55) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL7358689 0.72 NTSR1 (0.67) NTSR1RORCALDH1A1HTT
SCHEMBL13139586 0.72 NTSR1 (0.57) NTSR1KDM4EALDH1A1MAPT
SCHEMBL7362873 0.72 RORC (0.44) RORCTSHRHSD17B10
SCHEMBL14876504 0.71 NTSR1 (0.57) NTSR1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL5161966 0.71 IDO1 (0.48) RORCKDM4EALDH1A1TSHRHTT
SCHEMBL8029435 0.71 ATM (0.53) RORCKDM4EALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed