SCHEMBL7361693

SCHEMBL7361693

CC#CCOc1ccc(S(=O)(=O)NCCC(=O)OC(C)(C)C)cc1

nearest known ligand 0.70

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 18/20 0.70
MMP13 P45452 14/20 0.70
MMP1 P03956 13/20 0.70
MMP9 P14780 12/20 0.70
MMP14 P50281 2/20 0.60
MMP2 P08253 2/20 0.60
MMP7 P09237 2/20 0.49
MMP8 P22894 2/20 0.49
ADAM10 O14672 1/20 0.49
ALDH1A1 P00352 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362962 0.84 ADAM17 (0.78) ADAM17MMP13MMP1MMP9MMP14
SCHEMBL3944045 0.82 ADAM17 (1.00) ADAM17MMP13MMP1MMP9MMP14
SCHEMBL1336491 0.80 ALDH1A1 (0.49) ADAM17MMP13MMP1MMP9MMP2
SCHEMBL8576412 0.79 ALDH1A1 (0.56) ALDH1A1
SCHEMBL7356913 0.79 ADAM17 (0.69) ADAM17MMP13MMP1MMP9MMP14
SCHEMBL8347959 0.78 LMNA (0.56) MMP13MMP1MMP9MMP2ALDH1A1
SCHEMBL19450347 0.78 SIGMAR1 (0.50) MMP13MMP1MMP9MMP14MMP2
SCHEMBL6630004 0.77 ADAM17 (0.55) ADAM17MMP13MMP1MMP9MMP14
SCHEMBL6501738 0.77 ADAM17 (0.77) ADAM17MMP13MMP1MMP9MMP14
SCHEMBL7673440 0.77 MEP1B (0.60) MMP13MMP9MMP14MMP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326516-B1 RHEUMATIC DISEASES; SEPSIS; ANTIULCER AGENTS AMERICAN CYANAMID COMPANY 2001-12-04 US disclosed
EP-1147078-A1 ACETYLENIC (BETA)-SULFONAMIDO AND PHOSPHINIC ACID AMIDE HYDROXAMIC ACID TACE INHIBITORS American Cyanamid Company (US) 2001-10-24 EP disclosed
WO-2000044711-A1 ACETYLENIC $G(b)-SULFONAMIDO AND PHOSPHINIC ACID AMIDE HYDROXAMIC ACID TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed