SCHEMBL7364092

SCHEMBL7364092

Nc1n[nH]cc1-c1ccco1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.47
ADORA2A P29274 6/20 0.44
ADORA1 P30542 6/20 0.44
ADORA2B P29275 3/20 0.44
SMARCA2 P51531 1/20 0.42
PBRM1 Q86U86 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
ALDH1A1 P00352 5/20 0.42
MAPT P10636 4/20 0.42
HSD17B10 Q99714 4/20 0.42
KDM4E B2RXH2 4/20 0.42
POLB P06746 3/20 0.42
BLM P54132 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
PKM P14618 2/20 0.42
ALOX15 P16050 2/20 0.42
CASP1 P29466 2/20 0.42
CASP7 P55210 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065232 0.74 ADORA1 (0.43) PDPK1ADORA2AADORA1ADORA2BSMARCA2
SCHEMBL7260786 0.70 POLB (0.52) PDPK1ADORA2AADORA1TAAR1ALDH1A1
SCHEMBL6003619 0.70 KDR (0.38) PDPK1ALDH1A1MAPTHSD17B10KDM4E
SCHEMBL28457537 0.69 ADORA2A (0.47) PDPK1ADORA2AADORA1ADORA2BSMARCA2
SCHEMBL625453 0.69 ALDH1A1 (0.47) ADORA2AADORA1ADORA2BSMARCA2PBRM1
SCHEMBL16600588 0.69 TAAR1 (0.50) PDPK1ADORA2AADORA1ADORA2BSMARCA2
SCHEMBL11624096 0.68 KDM4E (0.50) PDPK1ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL4008741 0.67 GAA (0.38) PDPK1ADORA2AADORA1ADORA2BALDH1A1
SCHEMBL397270 0.67 ALDH1A1 (0.52) PDPK1ADORA2AADORA1ADORA2BSMARCA2
SCHEMBL544598 0.67 MAP4K4 (0.48) SMARCA2PBRM1ALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed