SCHEMBL7365657

SCHEMBL7365657

O=C1NCC(CCC2CCN(CC3=Cc4ccccc4OC3)CC2)N1c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365852 0.80 ACHE (0.52) ACHE
SCHEMBL7365661 0.78 DRD2 (0.43) ACHE
SCHEMBL7366544 0.72 SIGMAR1 (0.61)
SCHEMBL7367469 0.72 GBA1 (0.41) SLC6A2SLC6A4SLC6A3
SCHEMBL10667389 0.71 PARP1 (0.49) LTA4H
SCHEMBL7438133 0.69 ALOX5 (0.43) ACHE
SCHEMBL14454753 0.68 HTR2C (0.46) LTA4H
SCHEMBL14454752 0.67 HTR2C (0.46) LTA4H
SCHEMBL11188819 0.65 MEN1 (0.34) SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL10834103 0.64 MEN1 (0.33) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997028157-A1 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed