SCHEMBL7366544

SCHEMBL7366544

O=C1CC(CN2CCC(CCC3CNC(=O)N3c3ccccc3)CC2)Oc2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.61
HTR1A P08908 1/20 0.61
ABCB1 P08183 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366546 0.78 SIGMAR1 (0.62) SIGMAR1HTR1AABCB1
SCHEMBL7365852 0.75 ACHE (0.52)
SCHEMBL7365657 0.72 ACHE (0.36)
SCHEMBL7367469 0.71 GBA1 (0.41)
SCHEMBL15818378 0.70 SIGMAR1 (0.54) SIGMAR1HTR1AABCB1
SCHEMBL3613001 0.66 ABCB1 (0.64) SIGMAR1HTR1AABCB1
SCHEMBL3400551 0.66 ABCB1 (0.73) SIGMAR1HTR1AABCB1
SCHEMBL3397762 0.65 ABCB1 (0.61) SIGMAR1HTR1AABCB1
SCHEMBL11385907 0.64 SIGMAR1 (0.56) SIGMAR1HTR1AABCB1
SCHEMBL30124157 0.63 ADRA2A (0.51) SIGMAR1HTR1AABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997028157-A1 NOVEL PIPERIDINE DERIVATIVES 4-SUBSTITUTED BY AN IMIDAZOLIDIN-2-ON-1-YL-ETHYL, TETRAHYDROPYRIMIDIN-2-ON-1-YL-ETHYL AND 1,3-DIAZEPIN-2-ON-1-YL-ETHYL GROUP, AND USE THEREOF AS α2-ADRENERGIC RECEPTOR ANTAGONISTS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed