SCHEMBL7365744

SCHEMBL7365744

O=C(c1[c]cccc1)c1ccccc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
CNR2 P34972 2/20 0.47
CTNNB1 P35222 3/20 0.41
WNT3A P56704 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PTGS1 P23219 1/20 0.38
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
MAPK14 Q16539 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
PPIA P62937 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28311762 0.86 CTSS (0.44) LMNAGAA
SCHEMBL746794 0.80 LMNA (0.64) LMNAGAACNR2CTNNB1WNT3A
SCHEMBL28815055 0.78 LMNA (0.62) LMNAGAACNR2CTNNB1WNT3A
SCHEMBL9712664 0.77 CES2 (0.50) LMNAGAACYP2C9CYP2C19
SCHEMBL143892 0.75 ALDH1A1 (0.38)
SCHEMBL4388656 0.75 LIG1 (0.48) LMNAGAASMN1; SMN2CYP2C19SLC6A2
SCHEMBL5687866 0.75 LMNA (0.50) LMNAGAACNR2CTNNB1WNT3A
SCHEMBL22533769 0.74 HPGD (0.41) GAASMN1; SMN2MAPK14CYP2C9
SCHEMBL28055406 0.74 MAPT (0.53) GAASMN1; SMN2
SCHEMBL3717986 0.73 GAA (0.56) LMNAGAACNR2CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6037367-A Substituted-pent-4-ynoic acids SMITHKLINE BEECHAM CORPORATION (US) 2000-03-14 US disclosed
EP-0827495-A4 SUBSTITUTED-PENT-4-YNOIC ACIDS SMITHKLINE BEECHAM CORP (US) 1998-11-04 EP disclosed
EP-0827495-A1 SUBSTITUTED-PENT-4-YNOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1998-03-11 EP disclosed
WO-1997003945-A1 SUBSTITUTED-PENT-4-YNOIC ACIDS SMITHKLINE BEECHAM CORPORATION (US) 1997-02-06 WO disclosed