SCHEMBL7366117

SCHEMBL7366117

O=C(Nc1ccc(-c2c[nH]c(=O)cn2)cc1)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 1/20 0.53
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
POLB P06746 3/20 0.52
MITF O75030 2/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
MAPT P10636 5/20 0.52
MAPK1 P28482 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
PTPN1 P18031 2/20 0.48
HTT P42858 1/20 0.48
PTPN6 P29350 1/20 0.48
PTPN11 Q06124 1/20 0.48
MMP2 P08253 2/20 0.48
MMP9 P14780 2/20 0.48
MMP8 P22894 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396951 0.87 KMT2A (0.62) MEN1KMT2APOLBNPC1RAB9A
SCHEMBL7398689 0.84 ALOX12 (0.46) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL7364055 0.84 RAB9A (0.48) MEN1KMT2APOLBNPC1RAB9A
SCHEMBL7398136 0.83 POLB (0.55) MEN1KMT2APOLBNPC1RAB9A
SCHEMBL7391714 0.83 PTPN1 (0.67) MEN1KMT2ANPC1RAB9AALDH1A1
Bromide SCHEMBL10730898 0.82 PTPN1 (0.65) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL7396608 0.82 GAA (0.56) KMT2APOLBRAB9AMAPK1SMN1; SMN2
SCHEMBL16367722 0.78 KMT2A (0.76) P4HTMMEN1KMT2APOLBMITF
SCHEMBL23898948 0.77 KMT2A (0.83) P4HTMMEN1KMT2APOLBMITF
SCHEMBL8572381 0.77 KMT2A (0.83) P4HTMMEN1KMT2APOLBMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4657906-A CARDIOVASCULAR DISORDERS SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1987-04-14 US disclosed
US-4556711-A CARDIOTONIC AGENTS SMITH KLINE & FRENCH LABORATORIES LTD. (US) 1985-12-03 US disclosed
EP-0096517-A2 Aryl pyrazinones SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-12-21 EP disclosed