SCHEMBL7368577

SCHEMBL7368577

CCc1c(-c2ccncc2)nc(-c2ccc(OC)cc2OC)n1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CYP1A1 P04798 5/20 0.42
CYP1B1 Q16678 5/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2E1 P05181 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP4B1 P13584 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP3A5 P20815 1/20 0.41
CYP2A7 P20853 1/20 0.41
CYP3A7 P24462 1/20 0.41
CYP2F1 P24903 1/20 0.41
CYP2C18 P33260 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP2J2 P51589 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365190 0.86 NPC1 (0.51) NPC1RAB9ACYP1A1CYP1B1CYP1A2
SCHEMBL7366322 0.80 ALDH1A1 (0.49) NPC1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL4133106 0.72 NPC1 (0.64) NPC1RAB9ACYP1A1CYP1B1CYP1A2
SCHEMBL7365842 0.72 TGFBR1 (0.70) NPC1RAB9ATGFBR1TEKMAPK14
SCHEMBL7370785 0.72 CYP3A4 (0.51) NPC1RAB9ACYP1A1CYP1B1CYP1A2
SCHEMBL7372813 0.70 TLR8 (0.35) NPC1RAB9ATGFBR1TEKSMN1; SMN2
SCHEMBL7369909 0.70 NPC1 (0.52) NPC1RAB9ATGFBR1TEKMAPK14
SCHEMBL7373114 0.69 TLR9 (0.43) NPC1RAB9ACYP1A1CYP1B1MEN1
SCHEMBL7370568 0.68 CYP3A4 (0.55) NPC1RAB9ACYP1A1CYP1B1CYP1A2
SCHEMBL6283374 0.66 CRHR1 (0.71) CYP1A1CYP1B1CYP1A2CYP3A4CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4822805-A ANTIINFLAMMATORY AGENTS, CARDIOTONIC AGENTS, ANTIPLATELET AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-04-18 US disclosed
EP-0257897-A1 Imidazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-03-02 EP disclosed