SCHEMBL7369216

SCHEMBL7369216

Nc1cc(CC(N)C(=O)c2nccs2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.46
GABRD O14764 2/20 0.46
GABRA1 P14867 2/20 0.46
GABRB1 P18505 2/20 0.46
GABRG2 P18507 2/20 0.46
GABRB3 P28472 2/20 0.46
GABRA5 P31644 2/20 0.46
GABRA3 P34903 2/20 0.46
GABRA2 P47869 2/20 0.46
GABRB2 P47870 2/20 0.46
GABRA4 P48169 2/20 0.46
GABRE P78334 2/20 0.46
GABRA6 Q16445 2/20 0.46
GABRG1 Q8N1C3 2/20 0.46
GABRG3 Q99928 2/20 0.46
GABRQ Q9UN88 2/20 0.46
CPB2 Q96IY4 1/20 0.42
ALDH1A1 P00352 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377583 0.87 GABRP (0.43) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7374711 0.82 ALDH1A1 (0.44) ALDH1A1PLA2G4ACES1CMA1RECQL
SCHEMBL7373291 0.81 PLA2G4A (0.40) ALDH1A1NOS3NOS1NOS2PLA2G4A
SCHEMBL7373902 0.80 LOXL2 (0.46) ALDH1A1PLA2G4ACES1CMA1PTGS1
SCHEMBL25354508 0.77 GABRP (0.60) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22775321 0.77 GABRP (0.60) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29604446 0.77 GABRP (0.60) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL14780595 0.77 GABRP (0.60) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7371771 0.75 CPB2 (0.39) CPB2ALDH1A1PLA2G4ACES1CMA1
SCHEMBL27699627 0.71 ALDH1A1 (0.50) ALDH1A1PLA2G4ACES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057314-A ANTICOAGULANTS BIOCHEM PHARMA INC. (CA) 2000-05-02 US disclosed
EP-0802916-A1 LOW MOLECULAR WEIGHT BICYCLIC THROMBIN INHIBITORS BIOCHEM PHARMA INC (CA) 1997-10-29 EP disclosed
WO-1996019483-A1 LOW MOLECULAR WEIGHT BICYCLIC THROMBIN INHIBITORS BIOCHEM PHARMA INC. (CA) 1996-06-27 WO disclosed