SCHEMBL7369405

SCHEMBL7369405

CCOC(=O)CN1CCN(S(=O)(=O)Cc2ccccc2)CCC1=O

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.62
TSHR P16473 2/20 0.62
CYP2C19 P33261 1/20 0.62
NPSR1 Q6W5P4 2/20 0.56
PKM P14618 2/20 0.56
ALDH1A1 P00352 5/20 0.49
HSD17B10 Q99714 2/20 0.49
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
KDM4E B2RXH2 1/20 0.47
HPGD P15428 2/20 0.46
RAB9A P51151 1/20 0.46
F2 P00734 1/20 0.44
F10 P00742 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400981 0.76 ALDH1A1 (0.48) GAATSHRNPSR1ALDH1A1MAPT
SCHEMBL9708708 0.75 GSK3A (0.49) GAATSHRCYP2C19NPSR1ALDH1A1
SCHEMBL7365043 0.73 KMT2A (0.52) GAATSHRCYP2C19NPSR1ALDH1A1
SCHEMBL7397071 0.73 TSHR (0.52) GAATSHRCYP2C19NPSR1PKM
SCHEMBL9708647 0.73 ALDH1A1 (0.51) CYP2C19NPSR1ALDH1A1KMT2AMEN1
SCHEMBL735675 0.71 TSHR (0.81) GAATSHRCYP2C19ALDH1A1KMT2A
SCHEMBL7368700 0.70 RAB9A (0.48) GAATSHRCYP2C19NPSR1ALDH1A1
SCHEMBL3912922 0.70 TSHR (0.69) GAATSHRCYP2C19NPSR1ALDH1A1
SCHEMBL7366693 0.70 TSHR (0.51) TSHRCYP2C19NPSR1ALDH1A1KMT2A
SCHEMBL668453 0.69 TSHR (0.56) TSHRALDH1A1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211183-B1 PIPERAZINE DERIVATIVE ANTICOAGULANTS; ANTIISCHEMIC AGENTS; CARDIOVASCULAR DISORDERS COR THERAPEUTICS, INC. 2001-04-03 US disclosed
EP-0975625-A1 SELECTIVE FACTOR Xa INHIBITORS COR THERAPEUTICS, INC. (US) 2000-02-02 EP disclosed
WO-1998046591-A1 SELECTIVE FACTOR Xa INHIBITORS COR THERAPEUTICS, INC. (US) 1998-10-22 WO disclosed