SCHEMBL7370613

SCHEMBL7370613

CCn1nc(-c2ccc(C(=O)O)cc2)c2cccnc2c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.52
PDE4B Q07343 2/20 0.49
RORC P51449 2/20 0.47
TBXAS1 P24557 1/20 0.47
PDE4A P27815 2/20 0.45
RAB9A P51151 1/20 0.44
TSHR P16473 2/20 0.44
ALOX15 P16050 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
TP53 P04637 1/20 0.42
KAT2B Q92831 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA1 P30542 1/20 0.42
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
F2RL3 Q96RI0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360999 0.91 HPGD (0.53) HPGDRORCPDE4ARAB9ATSHR
SCHEMBL7365898 0.91 PDE4B (0.49) HPGDPDE4BRORCTBXAS1PDE4A
SCHEMBL7361314 0.89 TBXAS1 (0.46) HPGDPDE4BTBXAS1PDE4ARAB9A
SCHEMBL7365662 0.87 HPGD (0.55) HPGDPDE4BTBXAS1PDE4ATSHR
SCHEMBL7367402 0.87 NCOA1 (0.46) HPGDTBXAS1RAB9ATSHRGAA
SCHEMBL7365466 0.86 ALDH1A1 (0.56) HPGDPDE4BRORCPDE4AALOX15
SCHEMBL7372162 0.85 RAB9A (0.51) PDE4BTBXAS1PDE4ARAB9APDE4C
SCHEMBL7368362 0.84 PDE4A (0.54) HPGDPDE4BRORCPDE4AALOX15
SCHEMBL7365028 0.82 KDM4E (0.50) HPGDPDE4BTBXAS1PDE4ATSHR
SCHEMBL7369488 0.81 HPGD (0.50) HPGDPDE4BPDE4ARAB9AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed