SCHEMBL7370627

SCHEMBL7370627

O=c1nnc(-c2cccc(Cl)c2)c2[nH]cccc1-2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.51
IDO1 P14902 6/20 0.45
NUDT1 P36639 1/20 0.42
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
NOTUM Q6P988 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.37
RCE1 Q9Y256 1/20 0.37
TDO2 P48775 1/20 0.37
KDM5B Q9UGL1 1/20 0.36
MAPK13 O15264 1/20 0.36
RAF1 P04049 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366344 0.84 MAOB (0.50) MAOBIDO1ALDH1A1CYP1A2HPGD
SCHEMBL7370353 0.81 MAOB (0.53) MAOBADORA2AADORA1NOTUMALDH1A1
SCHEMBL7362866 0.80 MEN1 (0.44) IDO1KDM4EALDH1A1KMT2A
SCHEMBL7412116 0.79 NUDT1 (0.47) MAOBIDO1NUDT1ADORA2AADORA1
SCHEMBL7365581 0.78 CDK8 (0.48) ALDH1A1HPGDKDM5B
SCHEMBL7369411 0.77 RAB9A (0.42) KDM4EALDH1A1CYP1A2HPGDKMT2A
SCHEMBL7364174 0.75 KDR (0.46) ADORA2AADORA1KDM4EALDH1A1KMT2A
SCHEMBL7360220 0.73 MAP2K4 (0.40) KDM4EALDH1A1CYP1A2HPGDKMT2A
SCHEMBL7368926 0.73 CDK4 (0.47) MAOBIDO1ADORA1KDM4EALDH1A1
SCHEMBL7367836 0.72 IKBKB (0.42) IKBKBCHUKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612321-B1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX INC (US) 1999-08-25 EP disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed