SCHEMBL7373365

SCHEMBL7373365

Cc1ncn(C)c1C(C)([O])C(N)=O

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.37
ALDH1A1 P00352 1/20 0.37
KDM4E B2RXH2 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
PKM P14618 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
KAT2B Q92831 1/20 0.32
PIM3 Q86V86 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15592685 0.73 LMNA (0.51) LMNAALDH1A1KDM4EADORA3PKM
SCHEMBL19797901 0.72 APOBEC3A (0.41) LMNAALDH1A1KDM4EADORA3PKM
SCHEMBL25562761 0.66 APOBEC3A (0.39) LMNAALDH1A1
SCHEMBL15601778 0.64 LMNA (0.46) LMNAALDH1A1KDM4EADORA3PKM
SCHEMBL12123617 0.64 ALDH1A1 (0.39) LMNAALDH1A1
SCHEMBL7375007 0.64 APOBEC3A (0.38) LMNAALDH1A1ADORA2B
SCHEMBL7378481 0.63 KDM4E (0.42) LMNAALDH1A1KDM4EPIM3PIM2
SCHEMBL7379327 0.62 MPO (0.34)
SCHEMBL23930918 0.62 GABRA1 (0.36) ALDH1A1
SCHEMBL7375008 0.62 PDE4A (0.35) LMNAKDM4EADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed