SCHEMBL7375393

SCHEMBL7375393

NN=CNc1cccc(C(=O)CNc2ccccc2CCC(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.43
KDM4E B2RXH2 1/20 0.39
AGTR1 P30556 1/20 0.39
RAB9A P51151 1/20 0.39
PTGER1 P34995 2/20 0.38
PTGER4 P35408 2/20 0.38
PTGER3 P43115 2/20 0.38
PTGER2 P43116 2/20 0.38
SIRT1 Q96EB6 1/20 0.37
KCNK3 O14649 1/20 0.37
KCNK9 Q9NPC2 1/20 0.37
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
FFAR1 O14842 5/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
ITGAV P06756 1/20 0.34
FFAR4 Q5NUL3 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375119 0.83 FFAR1 (0.47) AKR1C3PTGER3ITGB3ITGA2BFFAR1
SCHEMBL7520432 0.82 AKR1C3 (0.44) AKR1C3AGTR1RAB9AITGB3ITGA2B
SCHEMBL7377645 0.78 BCHE (0.49) HDAC6
SCHEMBL7380190 0.78 KCNK3 (0.46) KCNK3KCNK9ITGB3ITGA2BITGAV
SCHEMBL8369251 0.77 CASP3 (0.52) KDM4EKCNK3KCNK9
SCHEMBL8432521 0.76 ABCB11 (0.41) PTGER1PTGER4PTGER3PTGER2SIRT1
SCHEMBL7380359 0.76 KCNK3 (0.46) RAB9AKCNK3KCNK9ITGB3ITGA2B
SCHEMBL7373860 0.75 PTGER1 (0.44) PTGER1PTGER4PTGER3PTGER2KCNK3
SCHEMBL7380550 0.74 ITGB3 (0.43) KDM4EKCNK3KCNK9ITGB3ITGA2B
SCHEMBL8429208 0.74 SIRT1 (0.37) PTGER1PTGER4PTGER3PTGER2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed