SCHEMBL7388752

SCHEMBL7388752

CC(C)(C)C(=O)Oc1cccc(-c2nc3cc(Cl)ccc3[nH]2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
CHEK2 O96017 3/20 0.44
AMY1A P0DUB6 1/20 0.43
ALDH1A1 P00352 4/20 0.42
KMT2A Q03164 4/20 0.42
HPGD P15428 3/20 0.42
MEN1 O00255 3/20 0.42
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
FTO Q9C0B1 1/20 0.42
HDAC3 O15379 5/20 0.42
HDAC4 P56524 5/20 0.42
HDAC1 Q13547 5/20 0.42
HDAC7 Q8WUI4 5/20 0.42
HDAC2 Q92769 5/20 0.42
HDAC10 Q969S8 5/20 0.42
HDAC11 Q96DB2 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386703 0.87 CHEK2 (0.48) KDM4ECHEK2AMY1AALDH1A1KMT2A
SCHEMBL7402117 0.86 KDM4E (0.61) KDM4EALDH1A1KMT2AHPGDMEN1
SCHEMBL7396027 0.84 HPSE (0.49) KDM4ECHEK2AMY1AALDH1A1KMT2A
SCHEMBL7396372 0.83 RAB9A (0.53) CHEK2ALDH1A1KMT2AMEN1MAPT
SCHEMBL23758270 0.81 AURKA (0.55) KDM4EAMY1AALDH1A1KMT2AHPGD
SCHEMBL7388111 0.81 AMY1A (0.66) KDM4ECHEK2AMY1AALDH1A1KMT2A
SCHEMBL7398683 0.80 ALDH1A1 (0.49) KDM4ECHEK2ALDH1A1HPGDHSD17B10
SCHEMBL7392370 0.79 AMY1A (0.46) KDM4EAMY1AALDH1A1RAB9ANPC1
SCHEMBL7388362 0.76 KDM4E (0.44) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL3336441 0.76 KDM4E (0.59) KDM4EALDH1A1KMT2AHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP claimed
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO disclosed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed