SCHEMBL7396235

SCHEMBL7396235

CC1CCc2c(N)c(Cl)cc(C(=O)O)c2O1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 3/20 0.39
HTR3A P46098 2/20 0.39
HTR1A P08908 1/20 0.39
ADRA2C P18825 1/20 0.39
ACHE P22303 1/20 0.39
PTGS1 P23219 1/20 0.39
ADRA1A P35348 1/20 0.39
KCNH2 Q12809 1/20 0.39
PARP1 P09874 1/20 0.38
MAPT P10636 1/20 0.36
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35
HSD11B1 P28845 1/20 0.35
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326376 0.92 HSD11B1 (0.36) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL7430275 0.86 PARP1 (0.49) PARP1HSD11B1HPGD
SCHEMBL8500114 0.76 HTR4 (0.40) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL1502018 0.76 HTR4 (0.51) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL7436836 0.75 MAOA (0.35) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL7332629 0.74 HTR4 (0.41) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL5316552 0.73 HTR4 (0.47) HTR4HTR3AHTR3EHTR3BHTR3D
Hydrochloric Acid SCHEMBL7137041 0.73 HTR3A (0.54) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL7393687 0.73 HTR4 (0.74) HTR4HTR3AHTR1AADRA2CACHE
SCHEMBL5042504 0.72 PTGES (0.37) HTR4HTR3AMAPTHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502209-A SIDE EFFECT REDUCTION, GASTROINTESTINAL SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-03-26 US disclosed
EP-0691341-A1 Benzopyrancarboxamide derivatives, salt thereof, process for the preparation of same and use thereof SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-01-10 EP disclosed