SCHEMBL7398172

SCHEMBL7398172

CC(C)CCN(C[C@H](O)CCc1ccccc1)C(=O)NCC(C)C

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.54
LMNA P02545 1/20 0.49
PKM P14618 1/20 0.49
KMT2A Q03164 5/20 0.45
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 3/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.42
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
OPRM1 P35372 3/20 0.40
OPRD1 P41143 3/20 0.40
OPRK1 P41145 3/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7547811 0.84 LMNA (0.45) HPGDLMNAPKMKMT2AALDH1A1
SCHEMBL6427941 0.80 LAP3 (0.52) HPGDLMNAPKMKMT2AALDH1A1
SCHEMBL8577651 0.73 MEN1 (0.39) HPGDLMNAPKMKMT2AALDH1A1
SCHEMBL4394350 0.72 CASR (0.53) HPGDLMNAPKMKMT2AALDH1A1
SCHEMBL10778356 0.71 LPAR1 (0.52) LMNAPKMKMT2AALDH1A1MEN1
SCHEMBL28808203 0.71 HPGD (1.00) HPGDLMNAPKMKMT2AALDH1A1
SCHEMBL8502371 0.70 OPRK1 (0.48) KMT2AALDH1A1MEN1TSHROPRM1
SCHEMBL8773812 0.70 SMN1; SMN2 (0.44) SMN1; SMN2
SCHEMBL10076985 0.70 TSHR (0.51) HPGDLMNAPKMKMT2AALDH1A1
Bicarbonate SCHEMBL27892668 0.69 TSHR (0.59) HPGDLMNAPKMKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0735019-A2 Retroviral protease inhibitors MONSANTO COMPANY (US) 1996-10-02 EP disclosed
EP-0731088-A2 Retroviral protease inhibitors MONSANTO COMPANY (US) 1996-09-11 EP disclosed
US-5482947-A ENZYME INHIBITORS FOR HIV PROTEASE INHIBITION FROM UREA OR THIOUREA COMPOUNDS TALLEY JOHN J (US) 1996-01-09 US disclosed
WO-1993023368-A1 UREA-CONTAINING HYDROXYETHYLAMINE COMPOUNDS AS RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1993-11-25 WO disclosed
EP-0558603-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1993-09-08 EP disclosed
WO-1992008688-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed