SCHEMBL7406367

SCHEMBL7406367

C=C(C(N)=O)c1c[nH]c(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.32
ALDH1A1 P00352 1/20 0.31
KCNN4 O15554 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405033 0.82 KCNN4 (0.36) KMT2AHTTKCNN4
SCHEMBL1828996 0.82 KDM4E (0.39) MAPTKMT2AALDH1A1
SCHEMBL6821893 0.79 ALDH1A1 (0.37) MAPTKMT2AALDH1A1KCNN4
SCHEMBL1830315 0.75 KCNN4 (0.40) MAPTKMT2AHTTALDH1A1KCNN4
SCHEMBL10896790 0.73 L3MBTL1 (0.39) MAPTKMT2AHTT
SCHEMBL18065068 0.71 TRPM8 (0.36) KCNN4
SCHEMBL8370808 0.70 LCK (0.38) KMT2A
SCHEMBL6821626 0.70 RECQL (0.50) MAPTKMT2AHTTALDH1A1
SCHEMBL3827052 0.70 KCNN4 (0.33) MAPTKMT2AALDH1A1KCNN4
SCHEMBL7974226 0.70 KDM4E (0.44) MAPTKMT2AHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0969840-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2001-02-28 EP disclosed
EP-0969840-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2000-01-12 EP disclosed
WO-1998042342-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 1998-10-01 WO disclosed