SCHEMBL8370808

SCHEMBL8370808

O=C(c1ccsc1)c1c[nH]c(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.38
FYN P06241 1/20 0.38
DAO P14920 1/20 0.38
HPGD P15428 1/20 0.38
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
HSD11B1 P28845 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
GPR52 Q9Y2T5 1/20 0.33
HDAC1 Q13547 1/20 0.33
KMT2A Q03164 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1828996 0.77 KDM4E (0.39) HPGDKMT2A
SCHEMBL6821893 0.75 ALDH1A1 (0.37) HDAC1KMT2A
SCHEMBL1830315 0.71 KCNN4 (0.40) HPGDKMT2ANPC1RAB9A
SCHEMBL7713125 0.71 CYP11B2 (0.38) HSD17B14
SCHEMBL7406367 0.70 MAPT (0.33) KMT2A
SCHEMBL10896790 0.69 L3MBTL1 (0.39) HPGDCES2CES1ADORA2AADORA1
SCHEMBL9182841 0.68 NPC1 (0.31) CES1NPC1RAB9A
SCHEMBL7405033 0.68 KCNN4 (0.36) CES1KMT2A
SCHEMBL18065068 0.68 TRPM8 (0.36) CES1
SCHEMBL838599 0.67 LCK (0.61) LCKFYNDAOHPGDCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999051593-A1 4-THIONAPHTHYL-1H-IMIDAZOLES WITH ALPHA-2-ADRENERGIC ACTIVITY ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 1999-10-14 WO disclosed