SCHEMBL7407707

SCHEMBL7407707

C[C@H](NS(=O)(=O)c1ccc(-c2ccc(Br)cc2)cc1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 15/20 1.00
MMP3 P08254 13/20 1.00
MMP13 P45452 13/20 1.00
MMP1 P03956 12/20 1.00
MMP7 P09237 11/20 1.00
MMP9 P14780 11/20 1.00
ADAMTS4 O75173 3/20 0.77
MMP14 P50281 1/20 0.74
SLC1A3 P43003 1/20 0.56
SLC1A2 P43004 1/20 0.56
SLC1A1 P43005 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407715 1.00 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL4651862 0.87 ADAMTS4 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL1751961 0.87 ADAMTS4 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL7404078 0.85 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL4424095 0.85 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL4433724 0.85 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL14191408 0.85 MMP2 (0.74) MMP2MMP3MMP13MMP1MMP7
SCHEMBL19785143 0.82 MMP2 (0.69) MMP2MMP3MMP13MMP1MMP7
SCHEMBL7409462 0.81 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7
SCHEMBL7409456 0.81 MMP2 (1.00) MMP2MMP3MMP13MMP1MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901466-B1 BIPHENYLSULFONAMIDE MATRIX METALLOPROTEINASE INHIBITORS WARNER LAMBERT CO (US) 2001-10-31 EP claimed
CN-1310629-A Combined administration of ACAT and MMP inhibitors for the treatment of atherosclerotic lesions WARNER LAMBERT CO (US) 2001-08-29 CN claimed
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP claimed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO claimed
EP-0901466-A1 BIPHENYLSULFONAMIDE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-03-17 EP claimed
US-5756545-A ANTIARTHRITIC AGENTS; OSTEOPOROSIS WARNER-LAMBERT COMPANY (US) 1998-05-26 US claimed
WO-1997044315-A1 BIPHENYLSULFONAMIDE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1997-11-27 WO claimed
US-20080119513-A1 Sulfonamide Derivative Selectively Inhibiting Mmp-13 SHIONOGI & CO., LTD. (JP) 2008-05-22 US disclosed
EP-0901466-B1 BIPHENYLSULFONAMIDE MATRIX METALLOPROTEINASE INHIBITORS WARNER LAMBERT CO (US) 2001-10-31 EP disclosed
US-5756545-A ANTIARTHRITIC AGENTS; OSTEOPOROSIS WARNER-LAMBERT COMPANY (US) 1998-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119513-A1 Sulfonamide Derivative Selectively Inhibiting Mmp-13 MMP13, MMP3, MMP11 MMP2 10/4885MMP3 2/4885MMP13 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.