SCHEMBL7408148

SCHEMBL7408148

CC(C)CC(C(=O)NC(C=O)CC(=O)O)C(=O)NC(CCC(=O)O)C(=O)Nc1cccc(Oc2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 3/20 0.44
CASP1 P29466 5/20 0.43
CTNNB1 P35222 5/20 0.43
MMP2 P08253 2/20 0.41
MMP8 P22894 2/20 0.41
CTSB P07858 1/20 0.41
MMP10 P09238 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
MMP14 P50281 1/20 0.40
SIRT5 Q9NXA8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414049 0.94 CASP1 (0.40) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7412858 0.94 CASP1 (0.40) MMP3CASP1CTNNB1MMP8CTSB
SCHEMBL7411983 0.92 CTNNB1 (0.46) MMP3CASP1CTNNB1
SCHEMBL7410916 0.92 MMP3 (0.46) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7411854 0.92 CASP1 (0.42) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7452753 0.92 MMP3 (0.47) MMP3CASP1MMP2MMP8CTSB
SCHEMBL7409752 0.91 MMP3 (0.40) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7409822 0.91 CASP1 (0.46) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7403974 0.91 MEN1 (0.41) MMP3CASP1CTNNB1MMP2MMP8
SCHEMBL7404374 0.91 CASP1 (0.40) MMP3CASP1MMP8CTSBMMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed