SCHEMBL7404374

SCHEMBL7404374

CC(C)CC(C(=O)NC(C=O)CC(=O)O)C(=O)NC(CCC#N)C(=O)Nc1cccc(Oc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.40
CTSB P07858 1/20 0.39
EGLN2 Q96KS0 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
MMP8 P22894 1/20 0.37
MITF O75030 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
MMP3 P08254 2/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
CASP3 P42574 1/20 0.36
CASP7 P55210 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408148 0.91 MMP3 (0.44) CASP1CTSBMMP8MMP3MMP9
SCHEMBL7452753 0.89 MMP3 (0.47) CASP1CTSBMMP8MMP3MMP1
SCHEMBL7412858 0.89 CASP1 (0.40) CASP1CTSBMMP8MMP3CASP3
SCHEMBL7414049 0.89 CASP1 (0.40) CASP1CTSBMMP8MMP3CTSK
SCHEMBL7411854 0.86 CASP1 (0.42) CASP1CTSBMMP8MITFALDH1A1
SCHEMBL7410711 0.85 MMP8 (0.46) CASP1CTSBMMP8MMP3MMP9
SCHEMBL7404158 0.84 NPY5R (0.43) CASP1CTSBMITFALDH1A1POLB
SCHEMBL7411983 0.83 CTNNB1 (0.46) CASP1ALDH1A1MMP3
SCHEMBL7410916 0.83 MMP3 (0.46) CASP1CTSBMMP8MMP3MMP1
SCHEMBL7409752 0.83 MMP3 (0.40) CASP1CTSBMMP8MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed