SCHEMBL7414049

SCHEMBL7414049

COC(=O)CCC(NC(=O)C(CC(C)C)C(=O)NC(C=O)CC(=O)O)C(=O)Nc1cccc(Oc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 6/20 0.40
MMP3 P08254 2/20 0.40
MMP2 P08253 1/20 0.40
CTSB P07858 1/20 0.39
CTNNB1 P35222 5/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSK P43235 1/20 0.38
MMP8 P22894 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408148 0.94 MMP3 (0.44) CASP1MMP3MMP2CTSBCTNNB1
SCHEMBL7412858 0.92 CASP1 (0.40) CASP1MMP3CTSBCTNNB1MMP8
SCHEMBL7406281 0.91 HDAC4 (0.39) CASP1MMP3MMP2CTSBMEN1
SCHEMBL7411854 0.90 CASP1 (0.42) CASP1MMP3MMP2CTSBCTNNB1
SCHEMBL7452753 0.89 MMP3 (0.47) CASP1MMP3MMP2CTSBMMP8
SCHEMBL7404374 0.89 CASP1 (0.40) CASP1MMP3CTSBCTSKMMP8
SCHEMBL7410711 0.88 MMP8 (0.46) CASP1MMP3MMP2CTSBMMP8
SCHEMBL7411983 0.88 CTNNB1 (0.46) CASP1MMP3CTNNB1TSHR
SCHEMBL7409752 0.87 MMP3 (0.40) CASP1MMP3MMP2CTSBCTNNB1
SCHEMBL7410916 0.86 MMP3 (0.46) CASP1MMP3MMP2CTSBCTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed