SCHEMBL7412858

SCHEMBL7412858

CC(C)CC(C(=O)NC(C=O)CC(=O)O)C(=O)NC(CCC(N)=O)C(=O)Nc1cccc(Oc2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.40
CTSB P07858 1/20 0.39
CASP3 P42574 1/20 0.39
CASP4 P49662 1/20 0.39
CASP5 P51878 1/20 0.39
CASP9 P55211 1/20 0.39
CASP6 P55212 1/20 0.39
CASP8 Q14790 1/20 0.39
CASP10 Q92851 1/20 0.39
CTNNB1 P35222 1/20 0.39
PSMB5 P28074 2/20 0.39
MMP8 P22894 2/20 0.38
MMP3 P08254 1/20 0.38
PSMB2 P49721 1/20 0.38
LTA4H P09960 1/20 0.38
TASP1 Q9H6P5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408148 0.94 MMP3 (0.44) CASP1CTSBCTNNB1MMP8MMP3
SCHEMBL7414049 0.92 CASP1 (0.40) CASP1CTSBCTNNB1MMP8MMP3
SCHEMBL7411854 0.90 CASP1 (0.42) CASP1CTSBCASP3CASP6CASP8
SCHEMBL7452753 0.89 MMP3 (0.47) CASP1CTSBMMP8MMP3
SCHEMBL7404374 0.89 CASP1 (0.40) CASP1CTSBCASP3CASP6CASP8
SCHEMBL7410711 0.88 MMP8 (0.46) CASP1CTSBMMP8MMP3
SCHEMBL7411983 0.86 CTNNB1 (0.46) CASP1CTNNB1MMP3
SCHEMBL7410916 0.86 MMP3 (0.46) CASP1CTSBCASP3CTNNB1MMP8
SCHEMBL7409752 0.86 MMP3 (0.40) CASP1CTSBCASP3CASP6CASP8
SCHEMBL7403974 0.85 MEN1 (0.41) CASP1CTSBCTNNB1MMP8MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed