SCHEMBL7411983

SCHEMBL7411983

COc1cccc(NC(=O)C(CCC(=O)O)NC(=O)C(CC(C)C)C(=O)NC(C=O)CC(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 6/20 0.46
CCKBR P32239 2/20 0.45
TSHR P16473 1/20 0.44
MMP3 P08254 1/20 0.42
CASP1 P29466 4/20 0.42
ALDH1A1 P00352 1/20 0.41
HDAC1 Q13547 1/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408148 0.92 MMP3 (0.44) CTNNB1MMP3CASP1
SCHEMBL7414032 0.89 CASP1 (0.47) CTNNB1MMP3CASP1
SCHEMBL7403974 0.88 MEN1 (0.41) CTNNB1MMP3CASP1LMNA
SCHEMBL7414049 0.88 CASP1 (0.40) CTNNB1TSHRMMP3CASP1
SCHEMBL7411011 0.88 MMP3 (0.53) CTNNB1MMP3CASP1
SCHEMBL7412858 0.86 CASP1 (0.40) CTNNB1MMP3CASP1
SCHEMBL7411007 0.86 CASP1 (0.45) CTNNB1TSHRMMP3CASP1ALDH1A1
SCHEMBL7406317 0.86 MMP3 (0.48) CTNNB1MMP3CASP1
SCHEMBL7406513 0.86 MMP1 (0.42) CTNNB1TSHRALDH1A1HDAC1LMNA
SCHEMBL7410916 0.86 MMP3 (0.46) CTNNB1MMP3CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed