SCHEMBL7410028

SCHEMBL7410028

CCOC(=O)NCC(=O)c1cccc(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 3/20 0.52
NPC1 O15118 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
RAB9A P51151 3/20 0.52
ALDH1A1 P00352 2/20 0.52
MAPT P10636 1/20 0.52
CES2 O00748 1/20 0.51
CES1 P23141 1/20 0.51
MAPK1 P28482 1/20 0.51
HTT P42858 1/20 0.51
MMP13 P45452 1/20 0.50
POLB P06746 1/20 0.50
BLM P54132 1/20 0.50
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23014560 0.83 MTNR1A (0.56) MTNR1BNPC1SMN1; SMN2RAB9ACES2
SCHEMBL20524444 0.82 KMT2A (0.60) NPC1ALDH1A1MAPTMAPK1HTT
SCHEMBL7440403 0.82 MTNR1A (0.63) MTNR1BNPC1SMN1; SMN2RAB9ACES2
SCHEMBL21509796 0.82 CES2 (0.50) MTNR1BNPC1SMN1; SMN2RAB9ACES2
SCHEMBL382162 0.81 ALDH1A1 (0.56) NPC1SMN1; SMN2RAB9AALDH1A1MAPT
SCHEMBL10782158 0.81 KMT2A (0.54) NPC1SMN1; SMN2RAB9AALDH1A1MAPT
SCHEMBL3846489 0.79 CES2 (0.61) MTNR1BNPC1SMN1; SMN2RAB9ACES2
Methane SCHEMBL11375164 0.79 KMT2A (0.53) NPC1SMN1; SMN2RAB9AALDH1A1MAPT
SCHEMBL7028931 0.79 KMT2A (0.56) NPC1SMN1; SMN2RAB9AALDH1A1MAPT
SCHEMBL7413883 0.79 MAPT (0.55) SMN1; SMN2ALDH1A1MAPTMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0107398-B1 ORTHO SUBSTITUTED DIHYDROXY-2(1H)QUINAZOLINONE-1-ALKANOIC ACIDS ORTHO PHARMA CORP (US) 1988-06-08 EP disclosed
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed