SCHEMBL7440403

SCHEMBL7440403

COc1cccc(C(=O)CNC(C)=O)c1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.63
MTNR1B P49286 9/20 0.63
CES2 O00748 1/20 0.57
CES1 P23141 1/20 0.57
HSD11B1 P28845 1/20 0.56
MMP13 P45452 1/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
POLB P06746 1/20 0.55
BLM P54132 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PARP1 P09874 1/20 0.54
TSHR P16473 1/20 0.54
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
CHRM3 P20309 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23014560 0.85 MTNR1A (0.56) MTNR1AMTNR1BCES2CES1MMP13
SCHEMBL7433393 0.85 SMN1; SMN2 (0.56) MTNR1ANPC1RAB9APOLBSMN1; SMN2
SCHEMBL3846489 0.84 CES2 (0.61) MTNR1AMTNR1BCES2CES1HSD11B1
SCHEMBL1194055 0.84 MMP13 (0.58) CES2CES1MMP13NPC1RAB9A
SCHEMBL10480836 0.83 KDM4E (0.56) MTNR1AMTNR1BSMN1; SMN2TSHR
SCHEMBL30758862 0.83 CES2 (0.69) MTNR1AMTNR1BCES2CES1HSD11B1
SCHEMBL11248287 0.83 CES2 (0.69) MTNR1AMTNR1BCES2CES1HSD11B1
Hydrochloric Acid SCHEMBL15974464 0.83 CES2 (0.59) MTNR1AMTNR1BCES2CES1HSD11B1
Hydrochloric Acid SCHEMBL3849048 0.83 CES2 (0.59) MTNR1AMTNR1BCES2CES1HSD11B1
SCHEMBL7410028 0.82 MTNR1B (0.52) MTNR1AMTNR1BCES2CES1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558756-B 2-aryl-2, 3-dihydro-4 (1H) -quinolinone semicarbazone compound and application thereof 沈阳药科大学 2021-08-03 CN disclosed
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed