SCHEMBL7410136

SCHEMBL7410136

CC(C)CCN(C[C@H](O)CCc1ccccc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
POLB P06746 1/20 0.42
HDAC8 Q9BY41 1/20 0.41
RORC P51449 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
MMP2 P08253 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
KCNA5 P22460 1/20 0.39
PER2 O15055 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8773812 0.74 SMN1; SMN2 (0.44) KCNA5SMN1; SMN2
SCHEMBL8502371 0.70 OPRK1 (0.48) ALDH1A1POLBOPRM1OPRD1OPRK1
SCHEMBL7398172 0.69 HPGD (0.54) ALDH1A1CYP2C9CYP2C19LMNAPKM
SCHEMBL10771432 0.69 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C9CYP2C19POLB
SCHEMBL10076985 0.69 TSHR (0.51) ALDH1A1LMNAPKMMMP2MMP9
SCHEMBL26103333 0.69 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7547811 0.68 LMNA (0.45) ALDH1A1LMNAPKMMMP2OPRM1
SCHEMBL14131205 0.68 HDAC8 (0.67) ALDH1A1CYP1A2CYP2C9CYP2C19HDAC8
SCHEMBL7411356 0.68 SMN1; SMN2 (0.44) KCNA5SMN1; SMN2
SCHEMBL8535085 0.68 TSHR (0.40) ALDH1A1LMNAPKMMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776971-A Heterocyclecarbonyl amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors G.D. SEARLE & CO. (US) 1998-07-07 US disclosed
US-5756533-A ENZYME INHIBITORS FOR TREATMENT OF AIDS G.D. SEARLE & CO. (US) 1998-05-26 US disclosed