SCHEMBL7410463

SCHEMBL7410463

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2cc(F)c(Br)cc2F)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.38
ITGA2B P08514 10/20 0.38
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
F2 P00734 4/20 0.33
TMPRSS6 Q8IU80 4/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
NR3C1 P04150 1/20 0.32
ITGAV P06756 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7410456 0.90 ITGB3 (0.47) ITGB3ITGA2BCA12CA1CA2
SCHEMBL7414402 0.88 POLB (0.49) ITGB3ITGA2BPOLBMEN1KMT2A
SCHEMBL7418122 0.88 ITGB3 (0.50) ITGB3ITGA2B
SCHEMBL7414101 0.87 ITGB3 (0.40) ITGB3ITGA2BPOLBF2TMPRSS6
SCHEMBL7415735 0.86 F2 (0.38) ITGB3ITGA2BMEN1KMT2ACA12
SCHEMBL7412871 0.85 MEN1 (0.40) ITGB3ITGA2BPOLBMEN1KMT2A
SCHEMBL7415207 0.85 ITGB3 (0.50) ITGB3ITGA2BCA12CA1CA2
SCHEMBL7414232 0.85 ITGB3 (0.37) ITGB3ITGA2BF2TMPRSS6CYP3A4
SCHEMBL7412728 0.85 F2 (0.39) ITGB3ITGA2BCA12CA1CA2
SCHEMBL7417980 0.85 MEN1 (0.40) ITGB3ITGA2BPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed