SCHEMBL7414743

SCHEMBL7414743

CCOc1ccc(S(=O)(=O)c2ccccc2)cc1C

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.53
POLB P06746 2/20 0.53
ALDH1A1 P00352 5/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
MAPT P10636 2/20 0.51
KMT2A Q03164 4/20 0.49
LMNA P02545 1/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.46
MEN1 O00255 3/20 0.44
WDR5 P61964 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
HTR6 P50406 2/20 0.44
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44
SFRP1 Q8N474 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14176668 0.88 ALDH1A1 (0.58) HTTPOLBALDH1A1SMN1; SMN2KMT2A
SCHEMBL9662390 0.86 HTT (0.52) HTTPOLBALDH1A1SMN1; SMN2KMT2A
SCHEMBL8058697 0.84 HTR6 (0.46) POLBALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL7417562 0.81 TP53 (0.42) HTTPOLBALDH1A1SMN1; SMN2MAPT
SCHEMBL9659632 0.79 ALDH1A1 (0.50) HTTPOLBALDH1A1SMN1; SMN2MAPT
SCHEMBL1949836 0.79 HTT (0.57) HTTPOLBALDH1A1SMN1; SMN2MAPT
SCHEMBL7416443 0.79 MMP2 (0.47) ALDH1A1LMNAPTGDR2
SCHEMBL9659630 0.79 FFAR4 (0.53) SMN1; SMN2MAPTLMNATDP1
SCHEMBL8061989 0.77 HTR6 (0.45) HTTPOLBALDH1A1SMN1; SMN2MAPT
SCHEMBL20847652 0.76 MEN1 (0.66) HTTALDH1A1SMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163214-A1 GAMMA-KETOACID DIPEPTIDES AS INHIBITORS OF CASPASE-3 Merck Frosst Canada & Co. (CA) 2001-12-19 EP disclosed
US-6225288-B1 IMPLICATED IN MODULATING APOPTOSIS; TREATMENT OF:CARDIAC AND CEREBRAL ISCHEMIA/REPERFUSION INJURY, SPINAL CORD INJURY AND ORGAN DAMAGE DURING TRANSPLANTATION, CHRONIC NEURODEGENERATIVE DISEASES, IMMUNODEFICIENCY, DIABETES, ALOPECIA, AGING MERK FROSST CANADA & CO. (CA) 2001-05-01 US disclosed
WO-2000055127-A1 GAMMA-KETOACID DIPEPTIDES AS INHIBITORS OF CASPASE-3 MERCK FROSST CANADA & CO. (CA) 2000-09-21 WO disclosed